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48

抑制剂 & 化合物

2

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Cat. No. Product Name Target Signaling Pathways
T2688 LY310762

LY310762 HCl

5-HT Receptor GPCR/G Protein; Neuroscience
LY310762 是 5-HT1D 受体拮抗剂,Ki 为 249 nM。
T0472 Venlafaxine hydrochloride

Venlafaxine HCl,盐酸文拉法辛,Wy 45030 hydrochloride

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Venlafaxine hydrochloride (Wy 45030 hydrochloride) 是一种口服有效的 5-羟色胺 (5-HT)/去甲肾上腺素 (NE) 重摄取的双重抑制剂,具有抗抑郁活性。
T0482 Sertraline hydrochloride

Sertraline HCl,CP-51974-1 HCl,盐酸舍曲林

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Sertraline hydrochloride (Sertraline HCl) 是选择性 5- 羟色胺再吸收抑制剂类的抗抑郁剂,可用于多种疾病的研究,如重度抑郁症和强迫症。
T6232 Vilazodone Hydrochloride

盐酸维拉佐酮,SB659746A,EMD 68843,Vilazodone HCl

Others; 5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience; Others
Vilazodone Hydrochloride (EMD 68843) 是 5-HT1A 受体和特异性 5-羟色胺再摄取抑制剂(SSRI) 的部分激动剂,用于治疗重度抑郁症。
T21029 Norfluoxetine Hydrochloride

Norfluoxetine HCl,去甲氟西汀

Others Others
Norfluoxetine Hydrochloride (Norfluoxetine HCl) 是氟西汀的活性代谢物。氟西汀是一种抗抑郁药。
T1189 Milnacipran hydrochloride

盐酸米那普仑,Milnacipran HCl,Savella,Dalcipran

Serotonin Transporter; Norepinephrine Neuroscience
Milnacipran hydrochloride (Savella) 是一种5-羟色胺-去甲肾上腺素重吸收抑制剂(SNRI),可用于纤维肌痛的研究。
T1042 Granisetron hydrochloride

盐酸格拉司琼,BRL 43694A,Granisetron HCl

5-HT Receptor GPCR/G Protein; Neuroscience
Granisetron hydrochloride (Granisetron HCl) 是一种5-HT3受体拮抗剂,可作为化疗后止吐剂。
T0088 Urapidil hydrochloride

Urapidil HCl,盐酸乌拉地尔

5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Urapidil hydrochloride (Urapidil HCl) 是α1-肾上腺素受体拮抗剂和5-HT1A 受体激动剂。
T1069 Metoclopramide hydrochloride

盐酸甲氧氯普胺,Maxolon,Metoclopramide HCl

Dopamine Receptor; 5-HT Receptor; AChR GPCR/G Protein; Neuroscience
Metoclopramide hydrochloride (Metoclopramide HCl) 是可口服的5-HT3和多巴胺D2受体拮抗剂,IC50值分别为 308 和 483 nM,用于恶心呕吐、胃食管反流和胃轻瘫的研究。
T6655 SB-269970 hydrochloride

SB-269970A,SB269970 HCl

5-HT Receptor GPCR/G Protein; Neuroscience
SB-269970 hydrochloride (SB-269970A) 是 SB-269970 的盐酸盐形式,是一种 5-HT7 受体拮抗剂,pKi 值为 8.3,对其选择性比其他 5-HT 受体大于50倍多。
T6461 Dapoxetine hydrochloride

LY-210448,LY-210448 hydrochloride,Dapoxetine HCl,盐酸达泊西汀,Priligy

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Dapoxetine hydrochloride (LY-210448 hydrochloride) 是一种具有口服活性的、选择性的血清素再摄取 (serotonin reuptake) 抑制剂 (SSRI),可用于研究早泄 (PE) 。
T0450L Fluoxetine hydrochloride

Fluoxetine HCl,盐酸氟西汀,LY-110140,Lilly110140

5-HT Receptor; Serotonin Transporter; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Fluoxetine hydrochloride (Lilly110140) 是一种高度特异性血清素摄取抑制剂。它被用作抗抑郁药,并且通常比传统的抗抑郁药具有更可接受的副作用特征。
T1528 Azasetron hydrochloride

Y-25130 hydrochloride,Y-25130 HCl,盐酸阿扎司琼,Azasetron HCl

5-HT Receptor GPCR/G Protein; Neuroscience
Azasetron hydrochloride (Y-25130 HCl) 是一种苯甲酰胺的衍生物,是有效的、选择性的5-HT3受体拮抗剂,可用于化疗引起的恶心呕吐研究。
T2132 Buspirone hydrochloride

Buspirone HCl,盐酸丁螺环酮,Narol,Buspar

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Buspirone hydrochloride (Buspar) 是一种 5HT(1A) 受体激动剂,可用于研究广泛性焦虑症。
T6814 Cyproheptadine hydrochloride

Periactin hydrochloride,Anarexol,盐酸赛庚啶,Cyproheptadine HCl,Nuran

5-HT Receptor GPCR/G Protein; Neuroscience
Cyproheptadine hydrochloride (Periactin hydrochloride) 是一种 5-HT2A 受体拮抗剂,具有抗抑郁和抗血清素作用。它具有抗血小板活性,可用于血栓栓塞性疾病的研究。
T6602 Naratriptan hydrochloride

Naratriptan HCl,Amerge,Naramig,盐酸那拉曲坦,GR-85548A hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
Naratriptan hydrochloride (GR-85548A hydrochloride) 是一种5-HT1受体激动剂,有抗偏头疼特性。它还可以通过刺激三叉神经系统感觉神经末梢上的 5-HT1D/1B 受体来发挥其作用,从而减少促炎神经肽的释放。
T7941 Imipramine hydrochloride

盐酸丙咪嗪,Imipramine (hydrochloride),Tofranil,G 22355,Imipramine HCl,Melipramine

Serotonin Transporter Neuroscience
Imipramine hydrochloride (Imipramine HCl) 可抑制血清素转运蛋白,IC50=32 nM。它可阻止胰酶的易位,阻碍 MV 和外泌体的分泌。
T8382 Cariprazine hydrochloride

Cariprazine HCl,盐酸卡利拉嗪,RGH188 hydrochloride

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Cariprazine hydrochloride (RGH188 hydrochloride) 是一种抗精神病药物,是一种 D3 和 D2 受体部分激动剂,Ki 分别为 0.09 nM 和 0.5 nM,对5-HT(1A)受体有一定亲和力。
T1509 Cyclobenzaprine hydrochloride

盐酸环苯扎林,Cyclobenzaprine HCl,MK130 hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
Cyclobenzaprine hydrochloride (MK130 hydrochloride) 是一种具有抗抑郁活性的中枢作用肌肉松弛剂,可减少肌肉痉挛。
T1173 Tropisetron hydrochloride

SDZ-ICS 930,Tropisetron HCl,ICS 205-930,盐酸托烷司琼

5-HT Receptor GPCR/G Protein; Neuroscience
Tropisetron hydrochloride (Tropisetron HCl) 是5-HT3受体拮抗剂和α7-烟碱受体激动剂,具有抗恶心和止吐活性,对5-HT3受体的 IC50为70.1 nM。
T1735 Lurasidone hydrochloride

Lurasidone HCl,SM-13496 (Hydrochloride),盐酸鲁拉西酮,SM-13496

Dopamine Receptor; 5-HT Receptor; Norepinephrine GPCR/G Protein; Neuroscience
Lurasidone hydrochloride (Lurasidone HCl) 是多巴胺 D2和5-HT7的拮抗剂,IC50值分别为 1.68 和 0.495 nM,用于治疗精神分裂症和双相情感障碍。它也是5-HT1A 受体的部分激动剂,IC50值为 6.75 nM。
T1619 Trazodone hydrochloride

KB-831,盐酸曲唑酮,Trazodone HCl,AF-1161

5-HT Receptor; Adrenergic Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Trazodone hydrochloride (Trazodone HCl) 是5 羟色胺受体拮抗剂和重吸收抑制剂,用作抗抑郁药,可治疗失眠和焦虑。
T1471 Duloxetine hydrochloride

Duloxetine HCl,盐酸度洛西汀,LY-248686 hydrochloride,(S)-Duloxetine hydrochloride,LY-248686 HCl

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine GPCR/G Protein; Neuroscience
Duloxetine hydrochloride ((S)-Duloxetine hydrochloride) 是一种 5-羟色胺-去甲肾上腺素重吸收 (serotonin-norepinephrine reuptake) 抑制剂 (SNRI),Ki=4.6 nM,可用于广泛性焦虑症的研究。
T0678 Amitriptyline hydrochloride

Amitriptyline HCl,Tryptizol,盐酸阿米替林,Domical,Annoyltin

Trk receptor; Sigma receptor; 5-HT Receptor; Serotonin Transporter; Sodium Channel; Adrenergic Receptor; AChR; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience; Tyrosine Kinase/Adaptors
Amitriptyline hydrochloride (Annoyltin) 是血清素再摄取转运体和去甲肾上腺素再摄取转运体抑制剂,还与多巴胺再摄取转运体结合,其Ki 为 2.58 μM。它也抑制肾上腺素能受体、毒蕈碱受体、组胺受体、5-羟色胺受体。它是TrkA 和TrkA 受体的激动剂,具有强神经营养活性和有抗抑郁作用。
T22936 Idalopirdine Hydrochloride

Lu AE58054盐酸盐,Lu AE58054 Hydrochloride,Idalopirdine HCl

5-HT Receptor GPCR/G Protein; Neuroscience
Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) 是一种选择性的5-HT6 受体拮抗剂,Ki 为 0.83 nM。
T10142L p-Ethynylphenylalanine hydrochloride

4-Ethynyl-L-phenylalanine HCL,p-Ethynylphenylalanine hydrochloride(278605-15-5 free base)

Hydroxylase Metabolism
p-Ethynylphenylalanine hydrochloride (4-Ethynyl-L-phenylalanine HCL) 是一种高效的、可逆的、选择性的、竞争性的色氨酸羟化酶 (TPH) 抑制剂,其Ki=32.6 μM。
T6616 Ondansetron hydrochloride

SN 307,盐酸昂丹司琼,帕罗西汀杂质A,Ondansetron HCl,Emeset,GR 38032 HCl,NSC 665799,Zofran

5-HT Receptor GPCR/G Protein; Neuroscience
Ondansetron hydrochloride (Zofran) 是5-HT3受体的拮抗剂,可用作化疗后止吐剂。
T3046 BMY 7378 dihydrochloride

BMY7378 HCl

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
BMY 7378 dihydrochloride (BMY7378 HCl) 是选择性 α1D 肾上腺素受体拮抗剂,也是5-HT1A 受体部分激动剂。它同表达克隆大鼠 α1D-AR 的膜结合的亲和力 (Ki=2 nM)  是同克隆大鼠 α1A-AR (Ki=800 nM) 或仓鼠 α1B-AR (Ki=600 nM) 结合的亲和力 的100 以上。
T0255 Clomipramine hydrochloride

Clomipramine HCl,Anafranil,盐酸氯米帕明

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine; GST GPCR/G Protein; Neuroscience; oxidation-reduction
Clomipramine hydrochloride (Anafranil) 是一种5-羟色胺转运体(Ki:0.14 nM)、去甲肾上腺素转运体(Ki:54 nM)和多巴胺转运体(Ki:3 nM)阻断剂。
T1636 Paroxetine hydrochloride

Paroxetine HCl,BRL29060 hydrochloride,FG-7051,BRL29060A,盐酸帕罗西汀

5-HT Receptor; Serotonin Transporter; GRK; AChR; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Paroxetine hydrochloride (Paroxetine HCl) 是一种血清素摄取抑制剂,能抑制 GRK2 活性,IC50值为 14 μM。它可研究抑郁症。
T8136 Perospirone hydrochloride

Perospirone HCl,盐酸哌罗匹隆,SM-9018 hydrochloride

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Perospirone hydrochloride (Perospirone HCl) 是非典型的抗精神病剂,可用于精神分裂症的研究。它是可口服的5-HT2A 受体和多巴胺 D2受体的拮抗剂,也是5-HT1A 受体的部分激动剂。
T0031L Ziprasidone hydrochloride

盐酸齐拉西酮,齐拉西酮盐酸盐,CP-88059 hydrochloride,CP-88059,Ziprasidone HCl

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Ziprasidone hydrochloride (CP-88059 hydrochloride) 是一种联合 5-HT(5-羟色胺)和多巴胺受体拮抗剂,具有抗精神病活性的强效作用。它也是去甲肾上腺素再摄取抑制剂。
T21446 Rotigotine Hydrochloride

Rotigotine (Hydrochloride),N 0923,N-0924,Rotigotine HCl,盐酸罗替戈汀,N-0923,罗替戈汀盐酸盐

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Rotigotine Hydrochloride (N-0924) 是多巴胺受体激动剂,是5-HT1A 受体的部分激动剂,以及α2B-肾上腺素受体的拮抗剂,具有抗帕金森病活性。
T8690 Brexpiprazole HCl

OPC 34712 dihydrochloride

Others Others
Brexpiprazole HCl (OPC 34712 dihydrochloride) 是一种新型抗精神病药物。
T0204 Protriptyline hydrochloride

盐酸普罗替林,Protriptyline HCl

5-HT Receptor; AChE GPCR/G Protein; Neuroscience
Protriptyline hydrochloride (Protriptyline HCl) 是一种含有一个仲胺的三环结构抗抑郁试剂,可以用于抑郁和 ADHD 的相关研究。它使动物精力充沛起激励作用,并且有时用于嗜睡症的相关研究。
T6572 Lorcaserin HCl

5-HT Receptor GPCR/G Protein; Neuroscience
Lorcaserin HCl 是一种选择性血清素激动剂,被批准为减肥药。
T30901 Chlorphentermine HCl

Chlorphentermine HCl is a serotonin transport substrate.
T26768 Benanserin HCl

Benanserin Hydrochloride,BAS,Benanserin,Benzyl antiserotonin

Benanserin HCl is a serotonin antagonist. It causes psychotropic effects in humans.
T69905 Iferanserin HCl

Iferanserin HCl is a selective serotonin receptor antagonist.
T34359 Ro 3-5940 HCl

Ro 3 5940 HCl

Ro 3-5940 HCl is a psychoactive agent, increasing in production of serotonin in central nervous system tissue.
T34559 SC-53116

SC 53116 HCl,SC53116 HCl

SC-53116 HCl can increase the production of serotonin in central nervous system tissues and is a psychoactive agent.
T33864 PAL-545 HCl

PAL-545 Hydrochloride,PAL545 Hydrochloride,PAL 545 Hydrochloride

PAL-545 HCl is a type of releaser of dual dopamine-serotonin (DA/5-HT) .
T71045 FK-1052 HCl

FK-1052 HCl is a serotonin 3 & 4 dual receptor antagonist.
T19629 Indeloxazine hydrochloride

CI-874l,Indeloxazine HCl,YM 08054-1,Indeloxazine,CI 874,CI874l

Indeloxazine HCl acts as a serotonin releasing agent, norepinephrine reuptake inhibitor, and NMDA receptor antagonist. Indeloxazine hydrochloride is an antidepressant and cerebral activator. It has been found to enhance acetylcholine release in the rat fo
T26184 Seproxetine HCl

(S)-Norfluoxetine hydrochloride,Seproxetine hydrochloride,(S)-Desmethylfluoxetine Hydrochloride

Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.
T69579 Dothiepin HCl

Dothiepin HCl is a Tricyclic antidepressant (TCA), acting as a serotonin–norepinephrine reuptake inhibitor (SNRI) and also having other activities including antihistamine, antiadrenergic, antiserotonergic, anticholinergic, and sodium channel-blocking effects.
T27689 JNJ-7925476 HCl

JNJ-7925476,JNJ7925476,JNJ 7925476

JNJ-7925476 HCl is a triple monoamine uptake inhibitor. JNJ-7925476 Salt blocks the dopamine transporter (DAT), norepinephrine transporter (NET) and serotonin transporter (SERT) in the central nervous system. The ED(50) values for JNJ-7925476 occupancy of
T69129 Clozapine HCl

Clozapine HCl is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, and displays a unique pharmacological profile. Clozapine is a serotonin antagonist, with strong binding to 5-HT 2A/2C receptor subtype. It also displays strong affinity to several dopaminergic receptors, but shows only weak antagonism at the dopamine D2 receptor, a receptor commonly thought to modulate neuroleptic activity. Agranulocytosis is a ...

化合物

LY310762
Cat.No: T2688
Synonym: LY310762 HCl
Target: 5-HT Receptor
Venlafaxine hydrochloride
Cat.No: T0472
Synonym: Venlafaxine HCl,盐酸文拉法辛,Wy 45030 hydrochloride
Target: 5-HT Receptor, Serotonin Transporter
Sertraline hydrochloride
Cat.No: T0482
Synonym: Sertraline HCl,CP-51974-1 HCl,盐酸舍曲林
Target: 5-HT Receptor, Serotonin Transporter
Vilazodone Hydrochloride
Cat.No: T6232
Synonym: 盐酸维拉佐酮,SB659746A,EMD 68843,Vilazodone HCl
Target: Others, 5-HT Receptor, Serotonin Transporter
Norfluoxetine Hydrochloride
Cat.No: T21029
Synonym: Norfluoxetine HCl,去甲氟西汀
Target: Others
Milnacipran hydrochloride
Cat.No: T1189
Synonym: 盐酸米那普仑,Milnacipran HCl,Savella,Dalcipran
Target: Serotonin Transporter, Norepinephrine
Granisetron hydrochloride
Cat.No: T1042
Synonym: 盐酸格拉司琼,BRL 43694A,Granisetron HCl
Target: 5-HT Receptor
Urapidil hydrochloride
Cat.No: T0088
Synonym: Urapidil HCl,盐酸乌拉地尔
Target: 5-HT Receptor, Adrenergic Receptor
Metoclopramide hydrochloride
Cat.No: T1069
Synonym: 盐酸甲氧氯普胺,Maxolon,Metoclopramide HCl
Target: Dopamine Receptor, 5-HT Receptor, AChR
SB-269970 hydrochloride
Cat.No: T6655
Synonym: SB-269970A,SB269970 HCl
Target: 5-HT Receptor
Dapoxetine hydrochloride
Cat.No: T6461
Synonym: LY-210448,LY-210448 hydrochloride,Dapoxetine HCl,盐酸达泊西汀,Priligy
Target: 5-HT Receptor, Serotonin Transporter
Fluoxetine hydrochloride
Cat.No: T0450L
Synonym: Fluoxetine HCl,盐酸氟西汀,LY-110140,Lilly110140
Target: 5-HT Receptor, Serotonin Transporter, Autophagy
Azasetron hydrochloride
Cat.No: T1528
Synonym: Y-25130 hydrochloride,Y-25130 HCl,盐酸阿扎司琼,Azasetron HCl
Target: 5-HT Receptor
Buspirone hydrochloride
Cat.No: T2132
Synonym: Buspirone HCl,盐酸丁螺环酮,Narol,Buspar
Target: Dopamine Receptor, 5-HT Receptor
Cyproheptadine hydrochloride
Cat.No: T6814
Synonym: Periactin hydrochloride,Anarexol,盐酸赛庚啶,Cyproheptadine HCl,Nuran
Target: 5-HT Receptor
Naratriptan hydrochloride
Cat.No: T6602
Synonym: Naratriptan HCl,Amerge,Naramig,盐酸那拉曲坦,GR-85548A hydrochloride
Target: 5-HT Receptor
Imipramine hydrochloride
Cat.No: T7941
Synonym: 盐酸丙咪嗪,Imipramine (hydrochloride),Tofranil,G 22355,Imipramine HCl,Melipramine
Target: Serotonin Transporter
Cariprazine hydrochloride
Cat.No: T8382
Synonym: Cariprazine HCl,盐酸卡利拉嗪,RGH188 hydrochloride
Target: Dopamine Receptor, 5-HT Receptor
Cyclobenzaprine hydrochloride
Cat.No: T1509
Synonym: 盐酸环苯扎林,Cyclobenzaprine HCl,MK130 hydrochloride
Target: 5-HT Receptor
Tropisetron hydrochloride
Cat.No: T1173
Synonym: SDZ-ICS 930,Tropisetron HCl,ICS 205-930,盐酸托烷司琼
Target: 5-HT Receptor
Lurasidone hydrochloride
Cat.No: T1735
Synonym: Lurasidone HCl,SM-13496 (Hydrochloride),盐酸鲁拉西酮,SM-13496
Target: Dopamine Receptor, 5-HT Receptor, Norepinephrine
Trazodone hydrochloride
Cat.No: T1619
Synonym: KB-831,盐酸曲唑酮,Trazodone HCl,AF-1161
Target: 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Duloxetine hydrochloride
Cat.No: T1471
Synonym: Duloxetine HCl,盐酸度洛西汀,LY-248686 hydrochloride,(S)-Duloxetine hydrochloride,LY-248686 HCl
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine
Amitriptyline hydrochloride
Cat.No: T0678
Synonym: Amitriptyline HCl,Tryptizol,盐酸阿米替林,Domical,Annoyltin
Target: Trk receptor, Sigma receptor, 5-HT Receptor, Serotonin Transporter, Sodium Channel, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor
Idalopirdine Hydrochloride
Cat.No: T22936
Synonym: Lu AE58054盐酸盐,Lu AE58054 Hydrochloride,Idalopirdine HCl
Target: 5-HT Receptor
p-Ethynylphenylalanine hydrochloride
Cat.No: T10142L
Synonym: 4-Ethynyl-L-phenylalanine HCL,p-Ethynylphenylalanine hydrochloride(278605-15-5 free base)
Target: Hydroxylase
Ondansetron hydrochloride
Cat.No: T6616
Synonym: SN 307,盐酸昂丹司琼,帕罗西汀杂质A,Ondansetron HCl,Emeset,GR 38032 HCl,NSC 665799,Zofran
Target: 5-HT Receptor
BMY 7378 dihydrochloride
Cat.No: T3046
Synonym: BMY7378 HCl
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Clomipramine hydrochloride
Cat.No: T0255
Synonym: Clomipramine HCl,Anafranil,盐酸氯米帕明
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine, GST
Paroxetine hydrochloride
Cat.No: T1636
Synonym: Paroxetine HCl,BRL29060 hydrochloride,FG-7051,BRL29060A,盐酸帕罗西汀
Target: 5-HT Receptor, Serotonin Transporter, GRK, AChR, Autophagy
Perospirone hydrochloride
Cat.No: T8136
Synonym: Perospirone HCl,盐酸哌罗匹隆,SM-9018 hydrochloride
Target: Dopamine Receptor, 5-HT Receptor
Ziprasidone hydrochloride
Cat.No: T0031L
Synonym: 盐酸齐拉西酮,齐拉西酮盐酸盐,CP-88059 hydrochloride,CP-88059,Ziprasidone HCl
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Norepinephrine, Histamine Receptor
Rotigotine Hydrochloride
Cat.No: T21446
Synonym: Rotigotine (Hydrochloride),N 0923,N-0924,Rotigotine HCl,盐酸罗替戈汀,N-0923,罗替戈汀盐酸盐
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Brexpiprazole HCl
Cat.No: T8690
Synonym: OPC 34712 dihydrochloride
Target: Others
Protriptyline hydrochloride
Cat.No: T0204
Synonym: 盐酸普罗替林,Protriptyline HCl
Target: 5-HT Receptor, AChE
Lorcaserin HCl
Cat.No: T6572
Synonym:
Target: 5-HT Receptor
Chlorphentermine HCl
Cat.No: T30901
Synonym:
Target:
Benanserin HCl
Cat.No: T26768
Synonym: Benanserin Hydrochloride,BAS,Benanserin,Benzyl antiserotonin
Target:
Iferanserin HCl
Cat.No: T69905
Synonym:
Target:
Ro 3-5940 HCl
Cat.No: T34359
Synonym: Ro 3 5940 HCl
Target:
SC-53116
Cat.No: T34559
Synonym: SC 53116 HCl,SC53116 HCl
Target:
PAL-545 HCl
Cat.No: T33864
Synonym: PAL-545 Hydrochloride,PAL545 Hydrochloride,PAL 545 Hydrochloride
Target:
FK-1052 HCl
Cat.No: T71045
Synonym:
Target:
Indeloxazine hydrochloride
Cat.No: T19629
Synonym: CI-874l,Indeloxazine HCl,YM 08054-1,Indeloxazine,CI 874,CI874l
Target:
Seproxetine HCl
Cat.No: T26184
Synonym: (S)-Norfluoxetine hydrochloride,Seproxetine hydrochloride,(S)-Desmethylfluoxetine Hydrochloride
Target:
Dothiepin HCl
Cat.No: T69579
Synonym:
Target:
JNJ-7925476 HCl
Cat.No: T27689
Synonym: JNJ-7925476,JNJ7925476,JNJ 7925476
Target:
Clozapine HCl
Cat.No: T69129
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2209 Serotonin hydrochloride

5-HT hydrochloride,5-羟基色胺盐酸盐,5-HT HCl,Serotonin HCl,5-Hydroxytryptamine hydrochloride

5-HT Receptor; Endogenous Metabolite; Transferase GPCR/G Protein; Metabolism; Neuroscience
Serotonin hydrochloride (Serotonin HCl) 是一种内源性 5-HT 受体激动剂、CNS 中的单胺神经递质和儿茶酚 O-甲基转移酶 (COMT) 抑制剂,Ki 值为 44 μM。
T1156 Palonosetron hydrochloride

盐酸帕洛诺司琼,RS 25259 197,Palonosetron HCl,RS 25259

5-HT Receptor GPCR/G Protein; Neuroscience
Palonosetron hydrochloride (RS 25259) 是一种 5-HT3 拮抗剂,用于预防和治疗化疗引起的恶心和呕吐。

天然产物

Serotonin hydrochloride
Cat.No: T2209
Synonym: 5-HT hydrochloride,5-羟基色胺盐酸盐,5-HT HCl,Serotonin HCl,5-Hydroxytryptamine hydrochloride
Target: 5-HT Receptor, Endogenous Metabolite, Transferase
Palonosetron hydrochloride
Cat.No: T1156
Synonym: 盐酸帕洛诺司琼,RS 25259 197,Palonosetron HCl,RS 25259
Target: 5-HT Receptor
TargetMol Loading
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